PKC-iota inhibitor 1

CAS No. 2328094-11-5

PKC-iota inhibitor 1( —— )

Catalog No. M22982 CAS No. 2328094-11-5

PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 147 Get Quote
5MG 219 Get Quote
10MG 349 Get Quote
25MG 583 Get Quote
50MG 833 Get Quote
100MG 1134 Get Quote
500MG 2268 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PKC-iota inhibitor 1
  • Note
    Research use only, not for human use.
  • Brief Description
    PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).
  • Description
    PKC-iota inhibitor 1 is an inhibitor of protein kinase C-iota (PKC-ι ; IC50 : 0.34 μM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PKC
  • Recptor
    PKC-ι
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2328094-11-5
  • Formula Weight
    374.4
  • Molecular Formula
    C21H22N6O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL?(333.83 mM;?Need ultrasonic)
  • SMILES
    O=C(C1=CC(C2=CC=CC(N3CCNCC3)=C2)=CN=C1N)NC4=CC=NC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kwiatkowski J, et al. Fragment-based Discovery of a Small-Molecule Protein Kinase C-iota Inhibitor Binding Post-kinase Domain Residues. ACS Med Chem Lett. 2019 Feb 15;10(3):318-323.
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